這本雜志的目的是發表對醫學化學和相關學科最新重要進展的簡短評論。藥物化學的小綜述范圍將涵蓋藥物化學的所有領域，包括合理藥物設計、合成化學、生物有機化學、高通量篩選、組合化學、藥物靶點以及天然產物研究和結構-活性關系研究的發展。《藥物化學小評》是每一位希望了解最新最重要進展的藥物和藥物化學家的重要刊物。

The aim of this journal is to publish short reviews on the important recent developments in medicinal chemistry and allied disciplines. The scope of Mini-Reviews in Medicinal Chemistry will cover all areas of medicinal chemistry including developments in rational drug design, synthetic chemistry, bioorganic chemistry, high-throughput screening, combinatorial chemistry, drug targets, and natural product research and structure-activity relationship studies. Mini-Reviews in Medicinal Chemistry is an essential journal for every medicinal and pharmaceutical chemist who wishes to be kept informed and up-to-date with the latest and most important developments.